医药中间体

重要中间体 Key Intermediates


Name
名称
Specification
标准
Imazalil sulfate
伊迈唑硫酸盐
In-house
Imazalil
伊迈唑碱
In-house
Alpha-(2,4-Dichlorophenyl)-1H-imidazol-1-ethanol
a-(2,4-二氯苯基)-1-氢咪唑-1-乙醇
In-house
(3-(Dimethylamino)propyl)triphenylphosphonium bromide hydrobromide (Olopatadine Hydrochloride Intermediate)
[3-(二甲基氨基)丙基]三苯基磷溴化物氢溴酸盐(盐酸奥洛他定中间体)
In-house
3-Methoxyfuran-2-carbaldehyde
3-甲氧基-2-呋喃醛
In-house
(4aS,8aS,9S)-3-(Benzyloxy)-4a-[(tert-butyldimethylsilyl)oxy]-9-(dimethylamino)-8a,9-dihydronaphtho[2,3-d]isoxazole-4,5(4aH,8H)-dione (Eravacycline Intermediate)
(4aS,8aS,9S)-3-(苄氧基)-4a-[(叔丁基二甲基硅基)氧基]-9-(二甲基氨基)-8a,9-二氢萘并[2,3-d]异噁唑-4,5(4aH,8H)-二酮(依拉环素中间体)
In-house
(S,E)-N-((3-(benzyloxy)isoxazol-5-yl)methylene)-2-methylpropane-2-sulfinamide (Eravacycline Intermediate K5)
(S,E)-N-((3-苄氧基异噁唑-5-基)亚甲基)-2-甲基丙烷-2-亚磺酰胺(依拉环素中间体K5)
In-house
(1S)-1-[3-(Benzyloxy)-1,2-oxazol-5-yl]-N,N-dimethylprop-2-en-1-amine L-(+)-tartrate (Eravacycline Intermediate K8)
(1S)-1-[3-(苄氧基)-1,2-噁唑-5-基]-N,N-二甲基丙-2-烯-1-氨基L-(+)-酒石酸盐(依拉环素中间体K8)
In-house

类固醇 API 及中间体 Steroids  APls&Intermediates


Name
名称
Specification
标准
Certificate
证书
Registration doc.
注册文件
Estradiol hemihydrate
雌二醇半水合物
EP / CP CEP / WC ASMF / DMF
Progesterone (un-micronized)
黄体酮(普粉)
EP / CP CEP ASMF
Progesterone (micronized)
黄体酮(微粉)
EP / CP CEP ASMF
Medrogestone
美屈孕酮
EP / /
Estrone
雌酚酮
In-house / /
Promestriene
普罗雌烯
In-house / /
Estradiol Valerate
戊酸雌二醇
EP / /
Estradiol benzoate
苯甲酸雌二醇
EP / CP / /


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